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標題: Highly Efficient Cul-catalyzed N-Arylation of Azaheterocycles with Aryl Iodides Using 1,1,1-Tris(hydroxymethyl)ethane as a Tridentate O-Donor Ligand: A Shorter Route to Toloxatone and Formal Synthesis of Linezolid
作者: Chen, H.H.
Huang, H.M.
Chen, S.C.
Chen, Y.J.
關鍵字: Copper;Cross-coupling;N-Arylation;Azaheterocycles;1,1,1-Tris(hydroxymethyl)ethane;nitrogen-containing heterocycles;cross-coupling reactions;c-n;bond;formation;heteroaryl halides;arylboronic acids;mild conditions;copper;imidazoles;3-aryl-2-oxooxazolidines
Project: Journal of the Chinese Chemical Society
期刊/報告no:: Journal of the Chinese Chemical Society, Volume 57, Issue 1, Page(s) 14-18.
An efficient copper-catalyzed N-arylation of azaheterocycles with aryl iodides using 1,1,1-tris(hydroxymethyl)ethane as a tridentates O-donor ligand has been accomplished in good to excellent yields. Moreover, this highly efficient catalyst system has been successfully demonstrated to one-step synthesis of toloxatone and a shorter route to formal synthesis of linezolid in good yields.
ISSN: 0009-4536
Appears in Collections:化學系所

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