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標題: Synthesis of optically active alpha-aminobenzolactam via an oxidative-cyclization reaction
作者: Chang, C.Y.
Yang, T.K.
關鍵字: growth-hormone secretagogue;inhibitors;phenylalanine;scaffolds
Project: Tetrahedron-Asymmetry
期刊/報告no:: Tetrahedron-Asymmetry, Volume 14, Issue 14, Page(s) 2081-2085.
A convergent pathway for the asymmetric synthesis of (-)-alpha-aminobenzolactam I is described. For the first time, the key intermediate N-methoxybenzolactam 8 was prepared from L-homophenylalanine ethyl ester hydrochloride (LHPE.HCl) 5 by employing an oxidative cyclization in the presence of trifluoroacetic acid (TFA). (C) 2003 Elsevier Science Ltd. All rights reserved.
ISSN: 0957-4166
DOI: 10.1016/s0957-4166(03)00408-7
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